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DW10075, a novel selective and small-molecule inhibitor of VEGFR, exhibits antitumor activities both in vitro and in vivo 期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 3, 页码: 398-407
作者:  Li, Meng-yuan;  Lv, Yong-cong;  Tong, Lin-jiang;  Peng, Ting;  Qu, Rong;  Zhang, Tao;  Sun, Yi-ming;  Chen, Yi;  Wei, Li-xin;  Geng, Mei-yu;  Duan, Wen-hu;  Xie, Hua;  Ding, Jian
收藏  |  浏览/下载:179/0  |  提交时间:2016/07/19
Dw10075  Vegf/vegf Receptor Inhibitor  Antitumor  Angiogenesis  U87-mg Human Glioblastoma  
Design, synthesis and biological evaluation of O-linked indoles as VEGFR-2 kinase inhibitors (I) 期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 9, 页码: 1165-1168
作者:  Gao, Guo-Rui;  Li, Meng-Yuan;  Tong, Lin-Jiang;  Wei, Li-Xin;  Ding, Jian;  Xie, Hua;  Duan, Wen-Hu
浏览  |  Adobe PDF(484Kb)  |  收藏  |  浏览/下载:256/63  |  提交时间:2015/12/17
Vegfr-2  Inhibitor  Indole  
Discovery of anilinopyrimidine-based naphthamide derivatives as potent VEGFR-2 inhibitors 期刊论文
MEDCHEMCOMM, 2015, 卷号: 6, 期号: 7, 页码: 1375-1380
作者:  Lv, Yongcong;  Li, Mengyuan;  Cao, Sufen;  Tong, Linjiang;  Peng, Ting;  Wei, Lixin;  Xie, Hua;  Ding, Jian;  Duan, Wenhu;  Xie, H (reprint author), Chinese Acad Sci, Div Antitumor Pharmacol, State Key Lab Drug Res, Shanghai Inst Mat Med, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China.
收藏  |  浏览/下载:152/0  |  提交时间:2015/12/17
Discovery of a New Series of Naphthamides as Potent VEGFR-2 Kinase Inhibitors 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 5, 期号: 5, 页码: 592-597
作者:  Lv, Yongcong;  Li, Mengyuan;  Liu, Ting;  Tong, Linjiang;  Peng, Ting;  Wei, Lixin;  Ding, Jian;  Xie, Hua;  Duan, Wenhu
浏览  |  Adobe PDF(2015Kb)  |  收藏  |  浏览/下载:457/128  |  提交时间:2014/12/19
Angiogenesis  Huvec  Inhibitor  Naphthamide  Vegfr-2